[CAS NO. 1197879-16-5] GPR4 antagonist 1

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PRODUCTS SPECIFICATIONS [1197879-16-5]

Catalog

HY-101536

Brand

MCE

CAS

1197879-16-5

MDL	MFCD18803646
Molecular Weight	431.62
Molecular Formula	C27H37N5
SMILES	CC1=C2C(N(CC3=CC=C(/C=C/CN4CCN(C(C)C)CC4)C=C3)C(CC)=N2)=NC(C)=C1

For research use only. We do not sell to patients.

GPR4 antagonist 1 is a GPR4 antagonist, with an IC ₅₀ of 189 nM.

IC50: 189 nM (GPR4) ^[1] .

Oil

Room temperature in continental US; may vary elsewhere.

In Vitro:

DMSO : 125 mg/mL ( 289.61 mM ; Need ultrasonic)

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Concentration Solvent Mass	1 mg	5 mg	10 mg

* Please refer to the solubility information to select the appropriate solvent.

In Vivo:

1.

Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

Solubility: ≥ 2.08 mg/mL (4.82 mM); Clear solution
2.

Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

Solubility: 2.08 mg/mL (4.82 mM); Suspended solution; Need ultrasonic
3.

Add each solvent one by one: 10% DMSO >> 90% corn oil

Solubility: ≥ 2.08 mg/mL (4.82 mM); Clear solution

* All of the co-solvents are available by MCE.