[CAS NO. 1439399-45-7] Glutaminase-IN-3
PRODUCTS SPECIFICATIONS [1439399-45-7]
DESCRIPTION [1439399-45-7]
Overview
| MDL | MFCD28411496 |
|---|---|
| Molecular Weight | 452.45 |
| Molecular Formula | C19H19F3N6O2S |
| SMILES | O=C(CC1=CC=CC(OC(F)(F)F)=C1)NC2=NN=C(CCCCC3=NN=C(N)S3)C=C2 |
Summary
Glutaminase-IN-3 (compound 657) is a potent glutaminase inhibitor with an IC 50 of 0.24 μM for Glutaminase 1 (GLS1). Glutaminase-IN-3 is extracted from patent WO2014089048A1, compound 657 [1] .
Appearance
Solid
Shipping
Room temperature in continental US; may vary elsewhere.
Storage
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
Solvent & Solubility
DMSO : 50 mg/mL ( 110.51 mM ; Need ultrasonic)
Stock Solutions
| Concentration Solvent Mass | 1 mg | 5 mg | 10 mg |
|---|
| 1 mM | 2.2102 mL | 11.0509 mL | 22.1019 mL |
| 5 mM | 0.4420 mL | 2.2102 mL | 4.4204 mL |
| 10 mM | 0.2210 mL | 1.1051 mL | 2.2102 mL |