[CAS NO. 151358-48-4]  DIM-C-pPhCO2Me

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PRODUCTS SPECIFICATIONS [151358-48-4]

Catalog
HY-112056
Brand
MCE
CAS
151358-48-4

DESCRIPTION [151358-48-4]

Overview

MDLMFCD31697720
Molecular Weight380.44
Molecular FormulaC25H20N2O2
SMILESCOC(C1=CC=C(C(C2=CNC3=C2C=CC=C3)C4=CNC5=C4C=CC=C5)C=C1)=O

For research use only. We do not sell to patients.

Summary

DIM-C-pPhCO2Me is a nuclear receptor 4A1 (NR4A1) antagonist [1] . Antineoplastic activity [1] .


IC50 & Target

Nuclear receptor 4A1 (NR4A1) [1]


Appearance

Solid


Shipping

Room temperature in continental US; may vary elsewhere.


Storage

Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month

Solvent & Solubility

In Vitro:

DMSO : ≥ 125 mg/mL ( 328.57 mM )

* "≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6285 mL 13.1427 mL 26.2854 mL
5 mM 0.5257 mL 2.6285 mL 5.2571 mL
10 mM 0.2629 mL 1.3143 mL 2.6285 mL
* Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

    Solubility: ≥ 2.08 mg/mL (5.47 mM); Clear solution

  • 2.

    Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.08 mg/mL (5.47 mM); Clear solution

* All of the co-solvents are available by MCE.


Synonyms

Benzoic acid, 4-(di-1H-indol-3-ylmethyl)-, methyl ester
Methyl 4-(di-1H-indol-3-ylmethyl)benzoate