[CAS NO. 2309668-44-6] DerazantinibRacemate

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PRODUCTS SPECIFICATIONS [2309668-44-6]

Catalog

HY-19981A

Brand

MCE

CAS

2309668-44-6

DESCRIPTION [2309668-44-6]

Overview

MDL	-
Molecular Weight	468.57
Molecular Formula	C29H29FN4O
SMILES	COCCNCCC1=CC(NC2=NC=C3CC(C4=CC=CC=C4F)C5=CC=CC=C5C3=N2)=CC=C1

For research use only. We do not sell to patients.

Summary

Derazantinib Racemate (ARQ-087 Racemate) is the racemate of Derazantinib. Derazantinib is an orally bioavailable, ATP competitive tyrosine kinase inhibitor; exhibits potent activity against FGFR1-3 chondrocytes with IC ₅₀ s of 4.5, 1.8, and 4.5 nM, respectively.

Appearance

Solid

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

Solvent & Solubility

In Vitro:

DMSO : 100 mg/mL ( 213.42 mM ; Need ultrasonic)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.1342 mL	10.6708 mL	21.3415 mL
5 mM	0.4268 mL	2.1342 mL	4.2683 mL
10 mM	0.2134 mL	1.0671 mL	2.1342 mL

* Please refer to the solubility information to select the appropriate solvent.