[CAS NO. 23142-01-0] Pentoxyverine citrate

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PRODUCTS SPECIFICATIONS [23142-01-0]

Catalog

HY-B1055

Brand

MCE

CAS

23142-01-0

DESCRIPTION [23142-01-0]

Overview

MDL	-
Molecular Weight	525.59
Molecular Formula	C26H39NO10
SMILES	O=C(C1(C2=CC=CC=C2)CCCC1)OCCOCCN(CC)CC.O=C(CC(C(O)=O)(O)CC(O)=O)O

For research use only. We do not sell to patients.

Summary

Carbetapentane citrate is a selective inhibitor of the cough, with mild atropine-like effect and local anesthesia effect.

Clinical Trial

NCT Number	Sponsor	Condition	Start Date	Phase
NCT02183649	Boehringer Ingelheim	Healthy	November 2009	Phase 1

Appearance

Solid

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

DMSO : ≥ 36 mg/mL ( 68.49 mM )

* "≥" means soluble, but saturation unknown.

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	1.9026 mL	9.5131 mL	19.0262 mL
5 mM	0.3805 mL	1.9026 mL	3.8052 mL
10 mM	0.1903 mL	0.9513 mL	1.9026 mL

* Please refer to the solubility information to select the appropriate solvent.

In Vivo:

1.

Add each solvent one by one: 10% DMSO >> 40% PEG300 >> 5% Tween-80 >> 45% saline

Solubility: ≥ 2.08 mg/mL (3.96 mM); Clear solution
2.

Add each solvent one by one: 10% DMSO >> 90% (20% SBE-β-CD in saline)

Solubility: ≥ 2.08 mg/mL (3.96 mM); Clear solution
3.

Add each solvent one by one: 10% DMSO >> 90% corn oil

Solubility: ≥ 2.08 mg/mL (3.96 mM); Clear solution

* All of the co-solvents are available by MCE.

Synonyms

Cyclopentanecarboxylic acid, 1-phenyl-, 2-[2-(diethylamino)ethoxy]ethyl ester, 2-hydroxy-1,2,3-propanetricarboxylate (1:1)

Cyclopentanecarboxylic acid, 1-phenyl-, 2-[2-(diethylamino)ethoxy]ethyl ester citrate (1:1)

Toclase

Carbetapentane citrate

Sedotussin

Pentoxyverine citrate

Tosnore

Calnathal

Antees

Tuclase

Fustpentane

Pencal

Carbetane

Germapect

Cossym

UCB 2543

2-(2-(Diethylamino)ethoxy)ethyl 1-phenylcyclopentanecarboxylate 2-hydroxypropane-1,2,3-tricarboxylate