[CAS NO. 1013937-63-7]  VTP-27999 TFA

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PRODUCTS SPECIFICATIONS [1013937-63-7]

Catalog
SLK-S2488
Brand
Selleck
CAS
1013937-63-7

DESCRIPTION [1013937-63-7]

Overview

MDLMFCD20278230
Molecular Weight639.1
Molecular FormulaC28H42ClF3N4O7
SMILESO=C(N1CCC[C@@H]([C@@H](OCCNC(OC)=O)C2=CC=CC(Cl)=C2)C1)NC[C@@H](NC)C[C@@H]3COCCC3.O=C(C(F)(F)F)O

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

1 mg5 mg10 mg
1 mM1.5647 mL7.8235 mL15.6470 mL
5 mM0.3129 mL1.5647 mL3.1294 mL
10 mM0.1565 mL0.7824 mL1.5647 mL
50 mM0.0313 mL0.1565 mL0.3129 mL

Description

VTP-27999 TFA (VTP-27999 Trifluoroacetate, VTP-27999 2,2,2-trifluoroacetate) is an orally efficacious, selecitive alkyl amine inhibitor with IC50 of 0.47 nM for 0.3 nM of purified recombinant human renin.

Targets

Renin [1]
(Cell-free assay)
0.47 nM