[CAS NO. 1161002-05-6] G15 (GRB-G15)
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PRODUCTS SPECIFICATIONS [1161002-05-6]
Catalog
SLK-S6651
Brand
Selleck
CAS
1161002-05-6
DESCRIPTION [1161002-05-6]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 370.24 |
| Molecular Formula | C19H16BrNO2 |
| SMILES | - |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 2.7010 mL | 13.5048 mL | 27.0095 mL |
| 5 mM | 0.5402 mL | 2.7010 mL | 5.4019 mL |
| 10 mM | 0.2701 mL | 1.3505 mL | 2.7010 mL |
| 50 mM | 0.0540 mL | 0.2701 mL | 0.5402 mL |
Description
G15 is a cell-permeable high affinity and selective antagonist with an affinity of approximately 20 nM that displays no affinity for ERα and ERβ at concentrations up to 10 μM.
Targets
| GPER [1] |
In vitro
G15 inhibits GPER-mediated proliferation stimulated by 17β-estradiol (E2) in A549 and H1793 cell lines. G15 inhibits the response of GPER stimulated by E2 and G1 in A549 and H1793 cell lines.
References
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