[CAS NO. ]  CP2

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PRODUCTS SPECIFICATIONS

Catalog
SLK-S8601
Brand
Selleck
CAS
-

DESCRIPTION

Overview

MDL-
Molecular Weight2010.15
Molecular FormulaC92H120N24O26S
SMILES-

For research use only.

Storage

3 years,-20°C,powder
1 years,-80°C,in solvent

Shipping

Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)

Preparing Stock Solutions

1 mg5 mg10 mg
1 mM0.4975 mL2.4874 mL4.9748 mL
5 mM0.0995 mL0.4975 mL0.9950 mL
10 mM0.0497 mL0.2487 mL0.4975 mL
50 mM---

Description

CP2 is a cyclic peptide that inhibits the with IC50 values of 42 nM and 29 nM for and , respectively.

Targets

KDM4C [1]
(Cell-free assay)
KDM4A [1]
(Cell-free assay)
29 nM42 nM

In vitro

CP2 uniquely binds in the KDM4A substrate-binding pocket. It binds differently to, but competes with, histone substrates in the active site.