[CAS NO. 1262132-81-9] Enarodustat (JTZ-951)
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PRODUCTS SPECIFICATIONS [1262132-81-9]
Catalog
SLK-S9656
Brand
Selleck
CAS
1262132-81-9
DESCRIPTION [1262132-81-9]
Overview
| MDL | - |
|---|---|
| Molecular Weight | 340.33 |
| Molecular Formula | C17H16N4O4 |
| SMILES | O=C(O)CNC(C1=C(O)C=C(CCC2=CC=CC=C2)N3C1=NC=N3)=O |
For research use only.
Storage
3 years,-20°C,powder
1 years,-80°C,in solvent
1 years,-80°C,in solvent
Shipping
Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)
Preparing Stock Solutions
| 1 mg | 5 mg | 10 mg | |
| 1 mM | 2.9383 mL | 14.6916 mL | 29.3832 mL |
| 5 mM | 0.5877 mL | 2.9383 mL | 5.8766 mL |
| 10 mM | 0.2938 mL | 1.4692 mL | 2.9383 mL |
| 50 mM | 0.0588 mL | 0.2938 mL | 0.5877 mL |
Description
Enarodustat (JTZ-951) is a potent and orally active inhibitor with IC50 of 0.22 μM for PHD2 and EC50 of 5.7 μM for EPO release from Hep3B cells. Enarodustat has the potential for the treatment of renal anemia.
Targets
In vitro
Enarodustat (JTZ-951) inhibits PHD2 with IC50 of 0.22 μM and the EPO release from Hep3B cells with EC50 of 5.7 μM.
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